Target Details
| UniProt AC | O00238 |
|---|---|
| Gene Symbol | BMPR1B |
| Protein Name | Bone morphogenetic protein receptor type-1B |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF01064 (Activin_recp) PF07714 (PK_Tyr_Ser-Thr) PF08515 (TGF_beta_GS) |
Summary
- Multi-target molecules 82
- Clinical molecules 12
- Avg pChEMBL 6.85
KEGG Pathways (7)
Associated Diseases (3)
Active Molecules (82)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
OATHVDKMFZZHHN
|
9.5 | Kd | 9 | — | |
QQWUGDVOUVUTOY
|
9.1 | Kd | 231 | Yes | |
DKZYXHCYPUVGAF
|
8.7 | Kd | 112 | — | |
MFAQYJIYDMLAIM
|
8.7 | Kd | 130 | Yes | |
VAARYSWULJUGST
|
8.4 | Kd | 119 | Yes | |
CDOVNWNANFFLFJ
|
7.9 | IC50 | 10 | — | |
KVLSZJPFQDRDPI
|
7.8 | IC50 | 4 | — | |
XIFIYBGPRFRYNP
|
7.8 | IC50 | 4 | — | |
KVDFCDPSKGACEZ
|
7.7 | IC50 | 4 | — | |
LOLPPWBBNUVNQZ
|
7.7 | Kd | 97 | Yes | |
MQFUFNHTCJRLKW
|
7.7 | IC50 | 6 | — | |
AGMGRCAUAZCHPG
|
7.5 | IC50 | 5 | — | |
OUKYUETWWIPKQR
|
7.5 | Kd | 31 | Yes | |
PAHLIVNOHVHPBG
|
7.4 | IC50 | 6 | — | |
CNEUJSQUCXSRDD
|
7.4 | Kd | 7 | — | |
FFLJVBPCONQSQW
|
7.4 | IC50 | 8 | — | |
RUBWYYYEDDAWLB
|
7.4 | IC50 | 5 | — | |
JMIFGARJSWXZSH
|
7.3 | IC50 | 3 | — | |
UPBPVAZUFAXUAC
|
7.3 | IC50 | 6 | — | |
IEJPGJXAWUJROQ
|
7.3 | IC50 | 5 | — | |
ZBNZXTGUTAYRHI
|
7.3 | Kd | 102 | Yes | |
UQEFQNWFVJXGDE
|
7.3 | IC50 | 3 | — | |
FAOGJKJCGFIFLI
|
7.2 | IC50 | 6 | — | |
UIARLYUEJFELEN
|
7.2 | Kd | 289 | Yes | |
WCDLCPLAAKUJNY
|
7.2 | IC50 | 8 | — | |
RKBYYWVZFBATHQ
|
7.2 | IC50 | 12 | — | |
FHTCHCUICJOIGJ
|
7.1 | IC50 | 7 | — | |
RIWTUJFFSTVYPW
|
7.1 | IC50 | 6 | — | |
BBDGBGOVJPEFBT
|
7.0 | IC50 | 6 | — | |
IIYOBXCNRFSCBH
|
7.0 | IC50 | 8 | — | |
UXVFRKCJRULCNV
|
7.0 | IC50 | 4 | — | |
YYLKKYCXAOBSRM
|
6.9 | Kd | 191 | — | |
BZXHYPDAQAEAKY
|
6.9 | IC50 | 5 | — | |
JUUFLLKHNYWHKP
|
6.9 | Kd | 12 | — | |
WMTXIPYJYDISKM
|
6.9 | IC50 | 8 | — | |
UAHBMBZHEHEEAW
|
6.8 | IC50 | 4 | — | |
ROCFHKYAFOQDHC
|
6.8 | IC50 | 5 | — | |
HKSZLNNOFSGOKW
|
6.8 | Kd | 408 | — | |
LMNXBEZQGBWMMY
|
6.7 | IC50 | 3 | — | |
UBTPOMHEYRBEHT
|
6.7 | IC50 | 5 | — | |
XYIZJZFZXCURDK
|
6.7 | IC50 | 5 | — | |
ALKJNCZNEOTEMP
|
6.7 | Kd | 55 | — | |
SHWKNOUREYUNBF
|
6.7 | IC50 | 6 | — | |
ZBOSAPQCJDMZCV
|
6.7 | IC50 | 6 | — | |
KTEIFNKAUNYNJU
|
6.6 | Kd | 114 | — | |
YTUZELSDHUVEFM
|
6.6 | IC50 | 4 | — | |
XHBVYDAKJHETMP
|
6.6 | IC50 | 24 | Yes | |
UHTHHESEBZOYNR
|
6.6 | Kd | 66 | Yes | |
GGQCWUKLPMFTDA
|
6.6 | IC50 | 5 | — | |
WTMROIBZVGJXRP
|
6.6 | IC50 | 4 | — |