Target Details
| UniProt AC | O00222 |
|---|---|
| Gene Symbol | GRM8 |
| Protein Name | Metabotropic glutamate receptor 8 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00003 (7tm_3) PF01094 (ANF_receptor) PF07562 (NCD3G) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 7.41
KEGG Pathways (4)
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WHUUTDBJXJRKMK
|
8.2 | IC50 | 20 | — | |
DDOQBQRIEWHWBT
|
7.2 | Ki | 4 | — | |
VLZBRVJVCCNPRJ
|
6.8 | IC50 | 4 | — |