Target Details
| UniProt AC | O00187 |
|---|---|
| Gene Symbol | MASP2 |
| Protein Name | Mannan-binding lectin serine protease 2 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00431 (CUB) PF07645 (EGF_CA) PF00084 (Sushi) PF00089 (Trypsin) |
Summary
- Multi-target molecules 88
- Clinical molecules 0
- Avg pChEMBL 6.98
KEGG Pathways (3)
Associated Diseases (1)
Active Molecules (88)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
XLTYUGDCGVDFET
|
6.8 | IC50 | 2 | — | |
ABQVZCJNLDVWKU
|
6.8 | IC50 | 2 | — | |
AOAQHXJRMLOUMO
|
6.8 | IC50 | 2 | — | |
CBGFPANNXANARQ
|
6.8 | IC50 | 2 | — | |
HWOZDKSFOHXMEO
|
6.8 | IC50 | 2 | — | |
PKWDOQSFFJDCGG
|
6.8 | IC50 | 2 | — | |
ARHYJCIBJJPJKC
|
6.7 | IC50 | 2 | — | |
CKSDDOVOKAXVKT
|
6.7 | Ki | 2 | — | |
LQRNULOTICMUKB
|
6.7 | IC50 | 2 | — | |
UAOULRPJIWQLSW
|
6.7 | IC50 | 2 | — | |
LPCIMCKUQYOLHW
|
6.7 | IC50 | 2 | — | |
GBBHETVEIGXSEU
|
6.7 | IC50 | 2 | — | |
HOGGSRIACGZTNH
|
6.7 | IC50 | 2 | — | |
IVPAQGGXKCGQER
|
6.7 | IC50 | 2 | — | |
WCIVODVYBXIAJJ
|
6.7 | IC50 | 2 | — | |
BLDLDULDJCSLSE
|
6.6 | IC50 | 2 | — | |
UTPFWUXZFWERAZ
|
6.6 | IC50 | 2 | — | |
YISLGRHFFVCCJW
|
6.6 | IC50 | 2 | — | |
LSUNMDRGMHQVSD
|
6.6 | IC50 | 2 | — | |
NPFQNQFRUYKRGV
|
6.5 | IC50 | 2 | — | |
TVFKZXKUBIQDST
|
6.5 | IC50 | 2 | — | |
VXJCOSNOIGKGMK
|
6.5 | IC50 | 2 | — | |
TYBRKUUAQWJMTB
|
6.4 | IC50 | 2 | — | |
NEBWVLBJKPHQNN
|
6.4 | IC50 | 2 | — | |
IDVMEVVVGSMSQJ
|
6.4 | IC50 | 2 | — | |
VVGBUDHDUBJJKT
|
6.4 | Ki | 2 | — | |
DWTZCKFHDROKLX
|
6.3 | IC50 | 2 | — | |
FCSLGKRXKHPWHX
|
6.3 | IC50 | 2 | — | |
WKVMPJHCNMEHRP
|
6.2 | IC50 | 2 | — | |
IXDGTHUYXMFLSM
|
6.2 | IC50 | 2 | — | |
WCDPLKUCPLBBNW
|
6.2 | IC50 | 2 | — | |
XWHZDLQFXCNTJR
|
6.2 | IC50 | 2 | — | |
DEHCIFBSNHVAOI
|
6.1 | IC50 | 2 | — | |
LVXBFWIZZVQJOV
|
6.0 | IC50 | 2 | — | |
OISOSMYTNZZBTL
|
6.0 | IC50 | 2 | — | |
BLRSMKZTKVSCSY
|
6.0 | IC50 | 2 | — | |
NBAVTEBIKQMCNU
|
6.0 | IC50 | 2 | — | |
NYXNZEVNQDDYHJ
|
6.0 | IC50 | 2 | — |