Target Details
| UniProt AC | O00141 |
|---|---|
| Gene Symbol | SGK1 |
| Protein Name | Serine/threonine-protein kinase Sgk1 |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF00069 (Pkinase) PF00433 (Pkinase_C) |
Summary
- Multi-target molecules 34
- Clinical molecules 3
- Avg pChEMBL 6.98
KEGG Pathways (6)
Active Molecules (34)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
DDKHTWASHUKHLD
|
9.0 | IC50 | 2 | — | |
MBNNXCKHRKSGSU
|
8.5 | IC50 | 2 | — | |
VYIKAHZTFTUSJO
|
8.5 | IC50 | 3 | — | |
GDVRVPIXWXOKQO
|
8.3 | IC50 | 10 | — | |
HKSZLNNOFSGOKW
|
8.0 | IC50 | 408 | — | |
WVSBGSNVCDAMCF
|
7.9 | IC50 | 4 | — | |
QNABDSWBQJKBHK
|
7.6 | IC50 | 45 | — | |
PABLVBARXHFRFL
|
7.5 | Kd | 5 | — | |
KSFDVNIKNYXUIP
|
7.4 | IC50 | 3 | — | |
PGBYHFSGSTUFFN
|
7.3 | IC50 | 2 | — | |
CZIVUSJISIAXJB
|
7.2 | IC50 | 18 | — | |
UEFCSGDOOJJXTN
|
7.2 | IC50 | 46 | — | |
CXSQMXRQOZZFLD
|
7.0 | IC50 | 18 | — | |
FXLKAGSPCQYANT
|
6.9 | IC50 | 2 | — | |
SXDPQGRNHSLZPC
|
6.8 | IC50 | 18 | — | |
XHIDFQRLXPJUMB
|
6.8 | IC50 | 2 | — | |
LYADGAGFYYXXIO
|
6.7 | IC50 | 82 | — | |
QKKIWEILHCXECO
|
6.7 | IC50 | 24 | — | |
AXTAPYRUEKNRBA
|
6.7 | IC50 | 24 | — | |
CZWJLLBPWLUINU
|
6.7 | IC50 | 10 | — | |
RTFQFPZKDYMMMJ
|
6.7 | IC50 | 2 | — | |
NDIUYMHNCUTVGE
|
6.6 | Ki | 25 | — | |
RAXZSEGXMBWYQK
|
6.6 | IC50 | 21 | — | |
MYHOUKHXSVKHBA
|
6.5 | IC50 | 3 | Yes | |
NXSJMRCTGYTSTK
|
6.5 | Kd | 200 | — | |
HBDSHCUSXQATPO
|
6.4 | IC50 | 14 | Yes | |
HOQNHSNBIIJJBO
|
6.4 | Ki | 7 | — | |
OSVUGUHRKMMBSE
|
6.2 | Kd | 170 | — | |
UJBJWYNPUOLFIZ
|
6.2 | IC50 | 49 | — | |
JPOSFPUHBHRUAX
|
6.2 | IC50 | 40 | Yes | |
YVQOYBIBWBAHKH
|
6.2 | IC50 | 12 | — | |
NGFGTMFVWSDFPS
|
6.1 | IC50 | 32 | — | |
IVVSBEQDCAZLFY
|
6.0 | IC50 | 333 | — | |
PALTUSLCLFDFQQ
|
6.0 | IC50 | 9 | — |