Target Details
| UniProt AC | E2QDN0 |
|---|---|
| Gene Symbol | thyA |
| Protein Name | Thymidylate synthase |
| Organism | Escherichia coli LF82 |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00303 (Thymidylat_synt) |
Summary
- Multi-target molecules 6
- Clinical molecules 3
- Avg pChEMBL 6.92
Active Molecules (6)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
GLRZVZIDWYADTN
|
7.8 | IC50 | 5 | Yes | |
BRVFNEZMTRVUGW
|
7.6 | IC50 | 3 | — | |
QPDXRVRRCIFNSL
|
7.3 | IC50 | 5 | Yes | |
DSIACOJIIGFHHZ
|
6.7 | IC50 | 4 | Yes | |
JJPUYFHYMITYSX
|
6.1 | IC50 | 2 | — | |
HWSZZBTVVLTRPO
|
6.1 | IC50 | 2 | — |