Target Details
| UniProt AC | D1MIX9 |
|---|---|
| Gene Symbol | blaGES-13 |
| Protein Name | beta-lactamase |
| Organism | Pseudomonas aeruginosa |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13354 (Beta-lactamase2) |
Summary
- Multi-target molecules 3
- Clinical molecules 0
- Avg pChEMBL 7.01
Top Co-occurrence Targets
- blaUOE-1 2 shared
- bla OXY 2 shared
- blaCTX-M-53 2 shared
- OXA-1 2 shared
- blaZ 2 shared
- blaSCO-1 2 shared
- KPC-2 1 shared
- blaTEM-1 1 shared
- blaTEM-125 1 shared
- 1 shared
Active Molecules (3)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
LPQZKKCYTLCDGQ
|
7.2 | IC50 | 15 | — | |
HZZVJAQRINQKSD
|
7.0 | IC50 | 13 | — | |
ZSKVGTPCRGIANV
|
6.8 | IC50 | 7 | — |