Target Details
UniProt ACC3SWJ7
Gene SymbolthyA
Protein NameThymidylate synthase
OrganismEscherichia coli
Entry Name
Organism Category Pathogen
Pfam Domains PF00303 (Thymidylat_synt)
Summary
  • Multi-target molecules 42
  • Clinical molecules 6
  • Avg pChEMBL 7.08
Top Co-occurrence Targets
Active Molecules (42)
InChIKey pChEMBL Type Targets Clinical
HTRZWDVKKNWTFT 9.5 Ki 2
ICKYKEQZWPNRNE 9.5 Ki 2
JFHSRPQQWWQYFB 8.8 Ki 2
PMTUUSDTAKQWQJ 8.3 Ki 2
KXIGHABTZWHJET 8.3 Ki 2
WDRLKIRDOFPOEI 8.1 Ki 2
HFEKDTCAMMOLQP 8.0 Ki 2
ZMOFGXPGBKVGSP 8.0 Ki 2
RSFXTHIRRXEJJD 7.8 IC50 5 Yes
LTKHPMDRMUCUEB 7.7 IC50 5 Yes
GOQIUYAAAGKJRE 7.6 Ki 2
ZTUSXMMVBQJSJX 7.4 Ki 2
SLCHNYIKJBZPFO 7.4 Ki 2
JOQXWQAZSGUWDV 7.4 IC50 6 Yes
YXHLVVWBIBKYIB 7.4 Ki 2
VFBJYFVJYIGZBN 7.4 Ki 2
MQXAYLIDIPHGSK 7.2 IC50 4 Yes
XHWRWCSCBDLOLM 7.1 Ki 2
OJMGRQBFCCRQMF 7.1 Ki 2
AIIOEPGQXVDMBH 6.8 Ki 2
KYXGMQCZCITEBX 6.8 Ki 2
RZPDNDSSUGJDEO 6.8 Ki 2
NDZXLRIRKARKDS 6.8 IC50 2
GTCLUWHIGIAUGO 6.6 IC50 2
NNJOOWYJGILHCE 6.5 Ki 3
MIISFGLDHJRHGS 6.5 IC50 2
MMVXYUMFIOTUHZ 6.5 Ki 2
SZWQFMKAPRFHLL 6.5 Ki 2
JXDJARWIPBCTJS 6.5 Ki 2
QDHQRSGEHWQARM 6.3 Ki 2
YMZRSTNMMRKKKX 6.3 Ki 2
HDVHULPVSPSYAG 6.3 Ki 2
PLRVFYBEWPHSDO 6.3 IC50 2
TXULAHBZZCHUNL 6.3 IC50 3 Yes
ARIQVZAPFSKYSS 6.2 IC50 2
GLAAJJXPUUQAKL 6.2 Ki 2
OJTJUBMLBHMYFG 6.2 Ki 2
QAWFAVXHJJBIED 6.2 Ki 2
BBSFBEFZYNIEPZ 6.2 Ki 2
JFDKEPQCKTUVRK 6.2 IC50 2
XEOQLLOHKNZVQZ 6.2 IC50 2
LTCOTSRHIWKZTK 6.1 IC50 3 Yes
2D structure