Target Details
| UniProt AC | B2RXH2 |
|---|---|
| Gene Symbol | KDM4E |
| Protein Name | Lysine-specific demethylase 4E |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF02373 (JmjC) PF02375 (JmjN) |
Summary
- Multi-target molecules 19
- Clinical molecules 0
- Avg pChEMBL 6.62
Active Molecules (19)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
WQXQGYTXHBAVJS
|
7.4 | IC50 | 4 | — | |
ZNWWSWJQMFNZDV
|
7.4 | IC50 | 5 | — | |
IDVBVEOFBRZZEI
|
7.3 | IC50 | 5 | — | |
DSGOLESVOJUGOK
|
7.0 | IC50 | 4 | — | |
OZMKCTFOIBLWOO
|
6.9 | IC50 | 5 | — | |
PSOBPHXKKHPWMU
|
6.8 | IC50 | 10 | — | |
XRMBRQWBOICYRP
|
6.7 | IC50 | 4 | — | |
JGRPKOGHYBAVMW
|
6.6 | IC50 | 13 | — | |
MJIVRKPEXXHNJT
|
6.5 | IC50 | 9 | — | |
YHHFKWKMXWRVTJ
|
6.5 | IC50 | 7 | — | |
AGEUQNZXCIVHPB
|
6.4 | IC50 | 2 | — | |
ARDXICZNEUJDDE
|
6.4 | IC50 | 5 | — | |
FRYSEKUUHUUJPX
|
6.4 | IC50 | 3 | — | |
PLQDLMAFBDRQSK
|
6.4 | IC50 | 4 | — | |
WUBIIGDBLTUSQG
|
6.4 | IC50 | 5 | — | |
IALMMJCSQDGXBB
|
6.3 | IC50 | 5 | — | |
ZTYRLXUTLYBVHH
|
6.3 | IC50 | 8 | — | |
YNQAUNMBAVKOIN
|
6.0 | IC50 | 2 | — | |
FDRUEUIWFFDWNQ
|
6.0 | IC50 | 2 | — |