Target Details
| UniProt AC | B0BL08 |
|---|---|
| Gene Symbol | dfrA17 |
| Protein Name | dihydrofolate reductase |
| Organism | Escherichia coli |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00186 (DHFR_1) |
Summary
- Multi-target molecules 223
- Clinical molecules 1
- Avg pChEMBL 7.55
Active Molecules (223)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
JGFFSKUMUVJYBC
|
6.3 | Ki | 2 | — | |
LFEJRVMXZUZEDH
|
6.3 | Ki | 2 | — | |
BJWZHTUBWSBYJS
|
6.2 | Ki | 2 | — | |
RNZGHILIUCETNY
|
6.2 | Ki | 3 | — | |
CBOOMIGGTVQYEO
|
6.2 | Ki | 2 | — | |
XOJSBWRVAWZFDY
|
6.2 | Ki | 2 | — | |
UTCUREXCXPTEBS
|
6.2 | Ki | 2 | — | |
AIZLSGCCJQCUJL
|
6.2 | Ki | 3 | — | |
VOFSSRGYMNQZKV
|
6.2 | IC50 | 2 | — | |
QQDUOWXAVYFFOJ
|
6.2 | Ki | 2 | — | |
XHPZVBGIPQQTQW
|
6.2 | Ki | 3 | — | |
IHTRXNSHXJVZTC
|
6.1 | Kd | 2 | — | |
LMZPSINLCOITEI
|
6.1 | IC50 | 3 | — | |
CJQWKDCPNDUIED
|
6.1 | IC50 | 2 | — | |
IHHWPKHCZVGDIM
|
6.1 | IC50 | 3 | — | |
OVBPIULPVIDEAO
|
6.1 | Kd | 2 | — | |
OUFZIPPLDRXXTA
|
6.1 | Ki | 2 | — | |
ZWQLWJWDJCCGFN
|
6.1 | Ki | 2 | — | |
GAYYBAJBQWLHKS
|
6.0 | IC50 | 3 | — | |
HAHWOBDKTAQBFE
|
6.0 | IC50 | 3 | — | |
NCLZDLNUFXETQQ
|
6.0 | Ki | 2 | — | |
VRXFDHXUFJMNEH
|
6.0 | Ki | 3 | — | |
IGTKNTAMQRRYRV
|
6.0 | IC50 | 3 | — |