Target Details
UniProt ACB0BL08
Gene SymboldfrA17
Protein Namedihydrofolate reductase
OrganismEscherichia coli
Entry Name
Organism Category Pathogen
Pfam Domains PF00186 (DHFR_1)
Summary
  • Multi-target molecules 223
  • Clinical molecules 1
  • Avg pChEMBL 7.55
Top Co-occurrence Targets
Active Molecules (223)
InChIKey pChEMBL Type Targets Clinical
AEVQGDTWXFVBNY 7.5 Ki 2
UADKZSUOVAPICX 7.5 Ki 2
VJXSSYDSOJBUAV 7.5 IC50 5
HPNCAZXFCHZMRO 7.4 Ki 2
UHUCUIUNKNVIKF 7.3 Ki 2
ALDCXILJAYAUTH 7.3 IC50 4
NBGMCAGDMQPEBF 7.3 Ki 2
LANUFFUDCPUKAX 7.2 Ki 2
NRJXHKNAIVZNNA 7.2 Ki 2
FSPRNSJDOJSXOP 7.2 Ki 2
LMMYDNOLGSNIBJ 7.2 Ki 2
FBLCVHLUKKJQGL 7.2 Ki 2
GKLNFRWZANFOPS 7.2 Ki 2
NNHKDVFXOLTUMW 7.2 Ki 2
BGGJCVGEWWWVHU 7.1 Ki 2
YGKDNGJMFQUDQL 7.0 Ki 2
VNYWLJDMMFVHSV 7.0 Ki 2
QYZVKLOHMLZHNF 7.0 Ki 2
ULJLXZHDPJDSAN 7.0 Ki 2
KUPCMNHSRONILW 7.0 IC50 3
PUMGLGGVAIIWCB 7.0 Ki 4
SUEPAWIBYITKPY 7.0 Ki 2
AKHBBXPUWYDYHT 7.0 Ki 2
FVXIRPQMUGBGDT 7.0 Ki 2
OXZQHMIUOCASIG 7.0 Ki 2
FXSZBFQPEMALCX 6.9 Ki 2
UZWIGXZSOSHNKZ 6.9 Ki 2
VJSZGADWCZOKOK 6.9 Ki 3
FKTRXRCVRZPVFR 6.9 Ki 2
GHEADESGVXHDFE 6.9 Ki 2
AWWRHLWEFOSBHS 6.9 Ki 2
CVKTUICDKSUYDI 6.9 IC50 3
IARRDWDIBSAXSX 6.9 Ki 2
OHYPUALOABANKC 6.9 Ki 2
ONRBLCNQZMSPEW 6.9 Ki 2
QROBKDOXPSLZLP 6.9 Ki 2
FBTWFHMLKCKSPR 6.9 Ki 3
JGWRJHQXTPUDRT 6.9 Ki 2
HZTFNSCZLJLPEO 6.8 IC50 4
VPSFLLCJENAQMF 6.8 IC50 3
QMRQJLSSCUTEQZ 6.8 Ki 2
FICBIZIKLGWVOK 6.8 Ki 2
HLGWCVIFHQFDSK 6.8 Ki 2
MBKGSXXZDBDJQC 6.8 Ki 2
NRQMIDHBGFQNEV 6.8 IC50 4
WHVMKGLHPRGZHK 6.8 Ki 3
YEWYWWJKFYYMNO 6.8 Ki 2
YMGUVTBVYOGUFZ 6.8 Ki 3
JOQXWQAZSGUWDV 6.7 IC50 6 Yes
RJFKHUXSEOMHCE 6.7 Ki 2
2D structure