Target Details
UniProt ACB0BL08
Gene SymboldfrA17
Protein Namedihydrofolate reductase
OrganismEscherichia coli
Entry Name
Organism Category Pathogen
Pfam Domains PF00186 (DHFR_1)
Summary
  • Multi-target molecules 223
  • Clinical molecules 1
  • Avg pChEMBL 7.55
Top Co-occurrence Targets
Active Molecules (223)
InChIKey pChEMBL Type Targets Clinical
ZKQGKWNKNGLJIB 8.6 Ki 2
UOELDAMKVYVBCC 8.6 Ki 2
YDMIFJZJSFJERI 8.6 Ki 2
KPUKMCAOBYZDQE 8.6 IC50 4
AHYITWBFECTSSJ 8.5 Ki 4
WWTCDGULAKAMHM 8.5 Ki 2
CHPPBLRQTGLSBZ 8.5 Ki 2
IEDVJHCEMCRBQM 8.4 Ki 7
SYIHNGNHJAJYQL 8.4 Ki 2
RNAWAVORHZUABK 8.4 Ki 2
HQXBYBOVCDPXCB 8.4 Ki 2
ORVQTLAPNXJUEJ 8.4 Ki 2
PETKLTZHTVYCPV 8.4 Ki 2
WSWJIZXMAUYHOE 8.3 Ki 2
ZUPNRVCYBHVECG 8.3 Ki 2
GMBNQAVADXFXRF 8.3 Ki 2
TUCQRMDCRDMAEG 8.3 IC50 4
VLQRVOAJCWFFQG 8.3 Ki 5
SZHHXYPKQHDKNL 8.2 Ki 3
VZTOIQAKDNEXFB 8.2 Ki 2
FBOZXECLQNJBKD 8.2 IC50 16
LMWNROFCHOPQFZ 8.2 Ki 3
YBJANOUTWRTBDK 8.1 IC50 4
DDNUPTARUMYNAL 8.1 IC50 4
DNDQAVBFTAVITN 8.0 Ki 2
WKSAUQYGYAYLPV 8.0 Ki 4
DPODCKRRIYULHE 8.0 Ki 2
HPOCGNHBIFZCAN 8.0 IC50 3
JCWCJLJGVCWEJH 8.0 Ki 2
YBIRDHJXPIORJB 7.9 Ki 3
OCUWNHFCHDFFHC 7.9 IC50 3
OTTAXGGOFALDRS 7.9 Ki 2
QABCVDFLEMLVBN 7.9 IC50 4
RCAKBZPOARPETR 7.9 Ki 2
ULAKSKJGSNQDHB 7.9 IC50 3
UQMGTQSCMRRWFV 7.9 Kd 2
SMHRXUOXEIKCBS 7.8 Ki 2
AAZRGUSAJLVIES 7.8 Ki 2
VUAPNJAVQJRKML 7.8 Ki 2
DWSNVSKRUMWIJX 7.8 Ki 2
RJRSBERDOBVYQI 7.8 IC50 2
RXNPBWYBFKJKIZ 7.7 Ki 2
LDBTVAXGKYIFHO 7.7 Ki 4
RZHLFYZKFQSTBC 7.7 Ki 2
GGYXPFIQXDUACT 7.7 Ki 2
SFSYDCBOGMLHHJ 7.7 Ki 2
WUZVJXBPZNLAIB 7.7 Ki 2
CJMXTBKLHYYCNQ 7.7 Ki 2
SCYCHUCWKNMIIH 7.7 Ki 2
CUEOPJOAMXKQSU 7.5 Ki 2
2D structure