Target Details
| UniProt AC | B0B3F0 |
|---|---|
| Gene Symbol | NS3/4A |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF01006 (HCV_NS4a) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 205
- Clinical molecules 0
- Avg pChEMBL 8.09
Active Molecules (205)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
MJXQFUHPNRVFRD
|
7.6 | IC50 | 4 | — | |
NSGBTQBHUVVQQK
|
7.6 | IC50 | 4 | — | |
RFBAMGIPTJOMSX
|
7.6 | IC50 | 4 | — | |
UOZVLIAVHBKHOK
|
7.6 | IC50 | 4 | — | |
YBTBVSQNDKHMPU
|
7.6 | IC50 | 4 | — | |
KHJUFJPLFNKMMO
|
7.5 | IC50 | 4 | — | |
PPLIHRDWIUFUOR
|
7.5 | IC50 | 4 | — | |
SFKSPKKZUGZHGG
|
7.5 | IC50 | 4 | — | |
VFFWWNSXYHEQFM
|
7.5 | IC50 | 4 | — | |
GHDPNYZUGAGWJK
|
7.5 | IC50 | 4 | — | |
KEYZYISKCGSJQI
|
7.5 | IC50 | 4 | — | |
LXTJVTZCNTYRMW
|
7.5 | IC50 | 4 | — | |
NAEFTBYPSLMAJV
|
7.5 | IC50 | 4 | — | |
QLSVUCOWXZXLOJ
|
7.5 | IC50 | 4 | — | |
AQILAUSZMZFFOH
|
7.4 | IC50 | 4 | — | |
AWQPGSZGZVXQPF
|
7.4 | Ki | 3 | — | |
LUULFVMVNHPTMD
|
7.4 | IC50 | 4 | — | |
RKSGIDSCASKYQC
|
7.4 | IC50 | 4 | — | |
SVIJSFDDCORCGI
|
7.4 | IC50 | 4 | — | |
VMGAVHOARRCARD
|
7.4 | IC50 | 4 | — | |
YAFHDFSMUJSRRC
|
7.4 | IC50 | 4 | — | |
ZGGFEFUZRQSHDM
|
7.4 | IC50 | 3 | — | |
KMRSRQTYTCFVAX
|
7.4 | Ki | 3 | — | |
LELTXNSBXZXYHC
|
7.3 | IC50 | 4 | — | |
NHNUZULGAZMHGX
|
7.3 | IC50 | 4 | — | |
OVLREHIDVJYZJD
|
7.3 | IC50 | 4 | — | |
ACYQAVZVIPDFCX
|
7.3 | IC50 | 4 | — | |
VWGQMMYCGJMUAB
|
7.3 | IC50 | 4 | — | |
XADSZCMEQSIZJY
|
7.2 | IC50 | 4 | — | |
RLWINPXRBXFVPF
|
7.2 | IC50 | 3 | — | |
DAQVNZCLEDKUSD
|
7.2 | IC50 | 4 | — | |
HUYACAOSSLGCFG
|
7.2 | IC50 | 4 | — | |
SBQMQLFREOTOLJ
|
7.2 | IC50 | 4 | — | |
TUGCYOIYHXSOKI
|
7.2 | IC50 | 4 | — | |
ZKELQISUOPVZIB
|
7.2 | IC50 | 4 | — | |
QANSKWRZMQTBLX
|
7.2 | IC50 | 4 | — | |
RBMZJAAUGKQFBX
|
7.2 | IC50 | 4 | — | |
XGAYJOVUJFIQOJ
|
7.2 | IC50 | 4 | — | |
DMXZRMUVJBHDST
|
7.1 | IC50 | 4 | — | |
PNJHHRKKKXJSKO
|
7.1 | IC50 | 4 | — | |
SKBNPHMFNYRNKO
|
7.1 | IC50 | 4 | — | |
UINMWOYMKDJTCK
|
7.0 | IC50 | 4 | — | |
VMGAVHOARRCARD
|
7.0 | IC50 | 4 | — | |
ZCDDKCMUQMFSAF
|
7.0 | IC50 | 4 | — | |
IRCSMPPIHNRCHT
|
7.0 | IC50 | 4 | — | |
HGAMFPMAHINILC
|
6.5 | IC50 | 4 | — | |
HTUQPKQGKVEYJP
|
6.4 | IC50 | 4 | — | |
RNFSHHKIOKRDGR
|
6.4 | IC50 | 4 | — | |
IVXYYGOHTXDSPQ
|
6.3 | IC50 | 4 | — | |
SFYGZRKQNXBACR
|
6.3 | IC50 | 4 | — |