Target Details
| UniProt AC | B0B3F0 |
|---|---|
| Gene Symbol | NS3/4A |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF01006 (HCV_NS4a) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 205
- Clinical molecules 0
- Avg pChEMBL 8.09
Active Molecules (205)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
SFPFFBUIHDKPII
|
8.2 | IC50 | 4 | — | |
BINCDYYXLHADFN
|
8.2 | IC50 | 4 | — | |
CKAFLNNMQJGEEX
|
8.2 | IC50 | 4 | — | |
PXWLCVOXAJCIHF
|
8.2 | IC50 | 4 | — | |
GCEYGBNIYJGZTN
|
8.2 | IC50 | 4 | — | |
LOKNAZXSPVVJPF
|
8.2 | IC50 | 4 | — | |
MVZJTRIKXSAMAF
|
8.2 | IC50 | 4 | — | |
SZDWNVOCTLNFPG
|
8.2 | IC50 | 4 | — | |
XNEUYKAPFWMJHA
|
8.2 | IC50 | 4 | — | |
BHALPSWCUUSMHK
|
8.1 | IC50 | 4 | — | |
DAXDBSLQHVZVKM
|
8.1 | IC50 | 4 | — | |
DJJPDGXKHXSURY
|
8.1 | IC50 | 4 | — | |
GCEYGBNIYJGZTN
|
8.1 | IC50 | 4 | — | |
GRLUHAWWANYLEN
|
8.1 | IC50 | 4 | — | |
JOSLQAAOZQRHRW
|
8.1 | IC50 | 4 | — | |
RDKJPYDNPLIEFF
|
8.1 | IC50 | 4 | — | |
RKPNCHNEDXAJST
|
8.1 | IC50 | 4 | — | |
ULLHRUAXAUBKJJ
|
8.1 | IC50 | 4 | — | |
VWXNOLOTOLRZRB
|
8.1 | IC50 | 4 | — | |
WCCYJARGTVUAAM
|
8.1 | IC50 | 4 | — | |
XSKKSWVGQBWSOZ
|
8.1 | IC50 | 4 | — | |
CUSGUKNSSJKVAE
|
8.1 | IC50 | 4 | — | |
GZMVTKDVGHBZSO
|
8.1 | IC50 | 4 | — | |
DAXDBSLQHVZVKM
|
8.0 | IC50 | 4 | — | |
JYCRVNJJDICZRJ
|
8.0 | IC50 | 4 | — | |
MSAOFHITMMVUMV
|
8.0 | IC50 | 4 | — | |
PWGWJCARSBIEBH
|
8.0 | IC50 | 4 | — | |
QBUJVJYBUBYHAE
|
8.0 | IC50 | 3 | — | |
RDHZGKIYONRFGL
|
8.0 | IC50 | 4 | — | |
SFBMHWHSTLMOCS
|
8.0 | IC50 | 3 | — | |
VNMXHBWOMGLDIH
|
8.0 | IC50 | 4 | — | |
WGQPESPJQGRZGU
|
8.0 | IC50 | 4 | — | |
XPKDLKMXYDYWGP
|
8.0 | IC50 | 4 | — | |
FSVNUGQYUJXOOG
|
8.0 | IC50 | 4 | — | |
IRJPOPFHQWLPAK
|
7.8 | IC50 | 3 | — | |
CFINSCMSFLQQAR
|
7.8 | IC50 | 4 | — | |
CMRUZHOEIPFESP
|
7.8 | IC50 | 4 | — | |
MMEBEYJGRMEXOT
|
7.8 | IC50 | 4 | — | |
SGHJJLBGKZIPSW
|
7.8 | IC50 | 4 | — | |
AFTKZUHBECRIPD
|
7.7 | IC50 | 4 | — | |
DTAGYFFAIVVJHG
|
7.7 | IC50 | 4 | — | |
JRBOXXSEYWPYMG
|
7.7 | IC50 | 4 | — | |
NAEFTBYPSLMAJV
|
7.7 | IC50 | 4 | — | |
QDLVNWRFJITDTF
|
7.7 | IC50 | 4 | — | |
QUTJDLPIJGFVTJ
|
7.7 | IC50 | 4 | — | |
UVNAIHPALNWIGA
|
7.7 | IC50 | 4 | — | |
XQWARQVHEJRBID
|
7.7 | IC50 | 4 | — | |
QFVVLWTXDCYIMN
|
7.7 | IC50 | 4 | — | |
BXZYHWGQDBDZKB
|
7.6 | IC50 | 4 | — | |
JFFCCDKBNGGOOE
|
7.6 | IC50 | 4 | — |