Target Details
| UniProt AC | B0B3F0 |
|---|---|
| Gene Symbol | NS3/4A |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF01006 (HCV_NS4a) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 205
- Clinical molecules 0
- Avg pChEMBL 8.09
Active Molecules (205)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RKNUBJJELTYQOF
|
8.6 | IC50 | 4 | — | |
SJNFJPFMHJLWNR
|
8.6 | IC50 | 4 | — | |
VNMXHBWOMGLDIH
|
8.6 | IC50 | 4 | — | |
DDZDRJQCCJHSJH
|
8.6 | IC50 | 4 | — | |
NALMWEJTNBTGFK
|
8.6 | IC50 | 4 | — | |
CFMGTKRBVVZVBF
|
8.5 | IC50 | 4 | — | |
HGMYODZJZPUWRC
|
8.5 | IC50 | 4 | — | |
HPKSTJTTXUFYNM
|
8.5 | IC50 | 4 | — | |
HQLIOGBJINMZFY
|
8.5 | IC50 | 4 | — | |
IQGJMNCUACIRBB
|
8.5 | IC50 | 4 | — | |
IWLXLASMFWNYHL
|
8.5 | IC50 | 4 | — | |
OALAYFQOTXVKEU
|
8.5 | IC50 | 4 | — | |
SSFQPBNIKXPGCC
|
8.5 | IC50 | 4 | — | |
ZZDPVPHOHNYTAU
|
8.5 | IC50 | 4 | — | |
RWXBAQMWNLSEBP
|
8.5 | IC50 | 4 | — | |
UTASHZYEMHIPHH
|
8.5 | IC50 | 3 | — | |
CTSWGNQIQFMNNJ
|
8.5 | IC50 | 4 | — | |
KCVVJXPLYSFXRJ
|
8.5 | IC50 | 4 | — | |
NJWQXXNLNZOZAW
|
8.5 | IC50 | 4 | — | |
RDHZGKIYONRFGL
|
8.5 | IC50 | 4 | — | |
RWXBAQMWNLSEBP
|
8.5 | IC50 | 4 | — | |
SJNFJPFMHJLWNR
|
8.5 | IC50 | 4 | — | |
XEPCTFXTGPAHEJ
|
8.5 | IC50 | 4 | — | |
QNRBXDCBCPJVRB
|
8.4 | IC50 | 3 | — | |
CFGJXJWENUPGMZ
|
8.4 | IC50 | 4 | — | |
RTDZYXVTDSBNJN
|
8.4 | IC50 | 4 | — | |
IAWKVVNKOOMFDE
|
8.4 | IC50 | 4 | — | |
GGDBDVHXMMLBAO
|
8.3 | IC50 | 4 | — | |
HBNQFHFXMNHZLQ
|
8.3 | IC50 | 4 | — | |
IQKDRVURUHCSRA
|
8.3 | IC50 | 4 | — | |
NLCBQIDOYIYGHS
|
8.3 | IC50 | 4 | — | |
PSDGVCIVPCWWSM
|
8.3 | IC50 | 4 | — | |
RDKJPYDNPLIEFF
|
8.3 | IC50 | 4 | — | |
RTBFYUQKYCYIGP
|
8.3 | IC50 | 4 | — | |
XEPCTFXTGPAHEJ
|
8.3 | IC50 | 4 | — | |
ZHBIJTQYLJKLSK
|
8.3 | IC50 | 4 | — | |
IQGJMNCUACIRBB
|
8.3 | IC50 | 4 | — | |
DGROTVCEUFXOSG
|
8.3 | Ki | 3 | — | |
MNXHOJWLGYZRKA
|
8.3 | IC50 | 4 | — | |
PEKAQWWCKOVJKE
|
8.3 | IC50 | 4 | — | |
QQHOKOMVWUCLCK
|
8.3 | IC50 | 4 | — | |
FDOUVNQZILTIRX
|
8.3 | IC50 | 3 | — | |
HLTMRTSTPMZYCW
|
8.3 | IC50 | 4 | — | |
ZEFCOSFYRNZVCT
|
8.3 | IC50 | 4 | — | |
BINCDYYXLHADFN
|
8.2 | IC50 | 4 | — | |
DLIOXULQASTBNO
|
8.2 | IC50 | 4 | — | |
DZNUXAJQSLZVLM
|
8.2 | IC50 | 4 | — | |
LUMMUNDAQFULAJ
|
8.2 | IC50 | 4 | — | |
NNTCLBUNHKJZRJ
|
8.2 | IC50 | 4 | — | |
OXYIGALIVPCFGR
|
8.2 | IC50 | 3 | — |