Target Details
| UniProt AC | B0B3F0 |
|---|---|
| Gene Symbol | NS3/4A |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF01006 (HCV_NS4a) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 205
- Clinical molecules 0
- Avg pChEMBL 8.09
Active Molecules (205)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
FSFUVODFJRFRKJ
|
10.0 | Ki | 3 | — | |
IHXGLDBKRROHDN
|
10.0 | Ki | 4 | — | |
NSICSOQWNRELKK
|
10.0 | Ki | 4 | — | |
NWXBVPNHAHFNDG
|
9.7 | Ki | 3 | — | |
CVFQOKIBZTWREC
|
9.6 | Ki | 4 | — | |
LYPMUUHUNIGEOB
|
9.5 | Ki | 4 | — | |
CFMGTKRBVVZVBF
|
9.3 | IC50 | 4 | — | |
JTZZSQYMACOLNN
|
9.3 | Ki | 6 | — | |
IQKDRVURUHCSRA
|
9.2 | IC50 | 4 | — | |
KRVBPGRPHRGDBE
|
9.2 | IC50 | 4 | — | |
ZIHXHTFVLKLWNX
|
9.2 | Ki | 4 | — | |
DMEMWXCZOKDOMY
|
9.1 | IC50 | 3 | — | |
IHPQWLFEUQBMFZ
|
9.1 | IC50 | 4 | — | |
KNQHCQDUNTWSPH
|
9.1 | IC50 | 4 | — | |
LOYIQGBTNJFCIL
|
9.1 | IC50 | 4 | — | |
NWFWLEAQCNXLAB
|
9.0 | IC50 | 4 | — | |
NWNRFJLJFPUJSR
|
9.0 | IC50 | 4 | — | |
OIHIJLNMNDCCIY
|
9.0 | IC50 | 4 | — | |
RZCUJQGMLLHXFG
|
9.0 | IC50 | 4 | — | |
WFXFHGMKTRFARM
|
9.0 | IC50 | 4 | — | |
YHJYFWRWHAHNQA
|
9.0 | IC50 | 4 | — | |
XLLUDKOBZFHIKN
|
8.9 | IC50 | 4 | — | |
XFYOTNPRWVBFPP
|
8.9 | IC50 | 4 | — | |
MOJHZLPPVIASCY
|
8.8 | IC50 | 4 | — | |
NLCBQIDOYIYGHS
|
8.8 | IC50 | 4 | — | |
VXDRIGYTIFAUHJ
|
8.8 | IC50 | 4 | — | |
YNYFVDOGUKBANE
|
8.8 | IC50 | 4 | — | |
AMWXBFDFQCGDLH
|
8.8 | IC50 | 4 | — | |
GNMJIFOVLJTJGQ
|
8.8 | IC50 | 4 | — | |
LRSKPOKZPAQFRH
|
8.8 | IC50 | 4 | — | |
VCYVRAYCTRSTDK
|
8.8 | IC50 | 4 | — | |
WXGVQUUZCZFRQM
|
8.8 | IC50 | 4 | — | |
CYWKRSLNXIMRQO
|
8.7 | IC50 | 4 | — | |
DBKVPPPOBUUZEG
|
8.7 | IC50 | 4 | — | |
GQEDTORABICPOM
|
8.7 | IC50 | 3 | — | |
GZPOQDPGYRPDKE
|
8.7 | IC50 | 4 | — | |
ILEXPDKMDMRQKR
|
8.7 | IC50 | 4 | — | |
OPNNEDOKBVIBDQ
|
8.7 | IC50 | 4 | — | |
RHEVGRYWYIGWAV
|
8.7 | IC50 | 4 | — | |
WFXFHGMKTRFARM
|
8.7 | IC50 | 4 | — | |
XONCCNBWLVICPL
|
8.7 | IC50 | 4 | — | |
XONCCNBWLVICPL
|
8.6 | IC50 | 4 | — | |
LTXGWCYRWMVHSW
|
8.6 | IC50 | 4 | — | |
XLMJBTKWBBMJFH
|
8.6 | Ki | 3 | — | |
CMGPWMKFYBSJKI
|
8.6 | IC50 | 4 | — | |
GGGMJNVXWGTZHR
|
8.6 | IC50 | 4 | — | |
HFIAXUYJXXCQEM
|
8.6 | IC50 | 4 | — | |
KNQHCQDUNTWSPH
|
8.6 | IC50 | 4 | — | |
OJIHYRADUMQJCL
|
8.6 | IC50 | 3 | — | |
QAKOEUGWCNOHLP
|
8.6 | IC50 | 4 | — |