Target Details
| UniProt AC | A9YLN7 |
|---|---|
| Gene Symbol | EML4/ALK fusion |
| Protein Name | Tyrosine-protein kinase receptor |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF07714 (PK_Tyr_Ser-Thr) |
Summary
- Multi-target molecules 7
- Clinical molecules 0
- Avg pChEMBL 8.56
Active Molecules (7)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PLCZCZWCIOPXGS
|
9.6 | IC50 | 3 | — | |
UMIDCBQSQODODG
|
9.6 | IC50 | 3 | — | |
KUKVPUVFVIDHDC
|
9.0 | IC50 | 3 | — | |
HLRNQALVSFYMKM
|
8.8 | IC50 | 3 | — | |
FMSDACLHKRTMHM
|
8.1 | IC50 | 3 | — | |
PWAFPCCSKIOXHE
|
7.8 | IC50 | 3 | — | |
FXGUUNXTWGWEDY
|
7.1 | IC50 | 3 | — |