Target Details
| UniProt AC | A9UEZ6 |
|---|---|
| Gene Symbol | BCR/ABL fusion |
| Protein Name | non-specific protein-tyrosine kinase |
| Organism | Homo sapiens |
| Entry Name | |
| Organism Category | Human |
| Pfam Domains | PF09036 (Bcr-Abl_Oligo) PF08919 (F_actin_bind) PF07714 (PK_Tyr_Ser-Thr) PF00621 (RhoGEF) PF00017 (SH2) |
Summary
- Multi-target molecules 5
- Clinical molecules 0
- Avg pChEMBL 6.85
Active Molecules (5)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
UKHOXYCPBAGGAN
|
7.3 | IC50 | 3 | — | |
YQXVNNKJNHKVLW
|
7.0 | IC50 | 3 | — | |
HWZFQQYDALNGQT
|
7.0 | IC50 | 3 | — | |
IQTSERMRWSERDI
|
6.8 | IC50 | 3 | — | |
MLAIONZVQZBMNT
|
6.1 | IC50 | 3 | — |