Target Details
UniProt ACA5X5Y0
Gene SymbolHTR3E
Protein Name5-hydroxytryptamine receptor 3E
OrganismHomo sapiens
Entry Name
Organism Category Human
Pfam Domains PF02931 (Neur_chan_LBD) PF02932 (Neur_chan_memb)
Summary
  • Multi-target molecules 183
  • Clinical molecules 6
  • Avg pChEMBL 7.84
Top Co-occurrence Targets
Active Molecules (183)
InChIKey pChEMBL Type Targets Clinical
FELGMEQIXOGIFQ 8.7 Kd 10
AASFRXJJHSMTFI 8.6 IC50 5
PEDIKBSWZVFPLW 8.6 IC50 5
ZGUGXTYWGBQHSU 8.6 Ki 5
HSLUKGWVBNRWNC 8.6 IC50 5
PDWZKMOQJPHUIY 8.6 Ki 5
NNRSVGLUJAPMQD 8.5 Ki 5
GZSKEXSLDPEFPT 8.5 Kd 5
CKUTYLGHNWXIJF 8.5 Ki 5
BLLXLUVDRGHQHD 8.5 IC50 5
APTTVZDGFWGGHT 8.4 Kd 5
HOMWNUXPSJQSSU 8.4 IC50 6
MPZDFMTUBDIVPH 8.4 IC50 5
OYASVWZGKNBLSA 8.3 IC50 5
CKXVQPZQTVVCCB 8.3 Kd 5
DNQOMGGYJRBLOX 8.3 Kd 5
PXNBOFBSFXZTES 8.3 Ki 5
RMKNXTZRZSDIHT 8.3 IC50 5
ZNRGQMMCGHDTEI 8.3 Kd 9
DXPJJGVPGVKFPQ 8.2 IC50 5
YQUHQGUROPITGF 8.2 Ki 5
XLVVGMWYXBVUJZ 8.2 Ki 5
ACSDLURGGYXLSE 8.2 IC50 5
VXYGXEFRVWLJIR 8.2 IC50 5
LJMASYWVOMQDML 8.2 IC50 5
KVDHVTQKKLVMJD 8.1 Ki 5
ZKSNSGVNASDNFY 8.1 Ki 5
MNJNPLVXBISNSX 8.1 IC50 5
SSQNUJKKRPIPQK 8.1 Kd 5
WZYBXWXOBIOGBH 8.1 Ki 5
BOHGZALGHLQJNA 8.0 IC50 7
ATJCEXDPRCAAOP 8.0 Ki 5
QENBLMVKRYFDIR 8.0 IC50 5
RDLIBCPWPNCFBW 7.9 Ki 5
XYOILXJZQNPSEP 7.9 IC50 7
ZJAWVBLMRPEUPW 7.9 Ki 5
JUSBDZIBILCYFG 7.9 IC50 5
SXXANLLRNHHDSR 7.8 IC50 5
XGEHMWGDEOZVML 7.8 IC50 5
AUISQHXDGNJFJZ 7.8 Ki 5
KQFRTJUIRPBBAB 7.8 Ki 5
DIHXJZHAIHGSAW 7.8 Ki 5
PXSRGUBKHGVLLK 7.7 Ki 5
BUOWEEIISDGZDM 7.7 IC50 5
ILDJOTZORZWBSP 7.7 IC50 5
AYDBLCSLKNTEJL 7.7 Kd 5
UNLXJJLVSBLRLU 7.7 Ki 5
YMQVTFAERCACRG 7.7 IC50 5
XGSROJUGJKXEPW 7.6 IC50 5
UVZMYAXDXQFDBO 7.6 IC50 5
2D structure