Target Details
| UniProt AC | A3FQ16 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | non-specific serine/threonine protein kinase |
| Organism | Cryptosporidium parvum (strain Iowa II) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 92
- Clinical molecules 6
- Avg pChEMBL 7.22
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KLNHTCQQONFNPS
|
7.0 | IC50 | 4 | — | |
XCFKTIVHIIOEHO
|
7.0 | IC50 | 4 | — | |
QGKJNBCCMVIKIT
|
7.0 | IC50 | 3 | — | |
OZTUULYOGSAFBT
|
6.9 | IC50 | 3 | — | |
WNSGCGVEGBFXSZ
|
6.9 | IC50 | 3 | — | |
YTTJKXSDNVYCBE
|
6.9 | IC50 | 3 | — | |
TYDGXGDYKRIRIF
|
6.9 | IC50 | 3 | — | |
GDQXJQSQYMMKRA
|
6.8 | IC50 | 15 | — | |
HUVZTPCJKNXREB
|
6.8 | IC50 | 5 | — | |
QFGDRGRJMYSRIW
|
6.8 | IC50 | 3 | — | |
HMRUGEAVJFRORJ
|
6.8 | IC50 | 3 | — | |
CJFWNLXLAAHQJY
|
6.8 | IC50 | 11 | Yes | |
GHQHPTZESKRASB
|
6.7 | IC50 | 3 | — | |
YJRWKOLRMSYZHE
|
6.7 | IC50 | 3 | — | |
UESYKRUJFLCOLW
|
6.7 | IC50 | 5 | — | |
IOMXIVABWISZJT
|
6.7 | IC50 | 3 | — | |
FOJGRLUYLZGTIX
|
6.6 | IC50 | 4 | — | |
PYEQRYTVMCYLNY
|
6.6 | IC50 | 4 | — | |
QKWPGKWGXYCSIM
|
6.6 | IC50 | 3 | — | |
FKNLUDCMGXLVRV
|
6.6 | IC50 | 4 | — | |
MGARWHQGMCYTAL
|
6.6 | IC50 | 4 | — | |
PNBDCDXPQZPIPK
|
6.5 | IC50 | 3 | — | |
TYGCWIRHRMMCNF
|
6.4 | IC50 | 3 | — | |
RGKPUWYSUXLERI
|
6.4 | IC50 | 3 | — | |
YHMLMIWKVKHAPH
|
6.4 | IC50 | 4 | — | |
DUPSNQFPAJUAKA
|
6.4 | IC50 | 9 | Yes | |
JHFJTTIYEGPPOW
|
6.4 | IC50 | 3 | — | |
SZRCRQLPOHAVJL
|
6.4 | IC50 | 3 | — | |
VPLRUYIVHZQYCE
|
6.2 | IC50 | 3 | — | |
XMTAJCWZZMFYID
|
6.2 | IC50 | 3 | — | |
KGLWFPORHQPXJI
|
6.2 | IC50 | 3 | — | |
QVMWSFYCPYOKBR
|
6.2 | IC50 | 3 | — | |
IXORERCONFMYQK
|
6.2 | IC50 | 3 | — | |
KAEFKAWNHDHBCY
|
6.2 | IC50 | 3 | — | |
MCKMGYSAHQYEDC
|
6.1 | IC50 | 3 | — | |
XNLZFVQIZBXQNM
|
6.1 | IC50 | 3 | — | |
TZDJIUGMUUUAQD
|
6.0 | IC50 | 3 | — | |
QAWHVZMZNTYGPK
|
6.0 | IC50 | 3 | — | |
QBINFJIYMSCWHV
|
6.0 | IC50 | 3 | — | |
YRYOEVHVROHLKR
|
6.0 | IC50 | 3 | — | |
DJAZYXTUKHPMNT
|
6.0 | IC50 | 3 | — | |
LMVAHLFZGWUGNF
|
6.0 | IC50 | 8 | Yes |