Target Details
| UniProt AC | A3FQ16 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | non-specific serine/threonine protein kinase |
| Organism | Cryptosporidium parvum (strain Iowa II) |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF13499 (EF-hand_7) PF00069 (Pkinase) |
Summary
- Multi-target molecules 92
- Clinical molecules 6
- Avg pChEMBL 7.22
Active Molecules (92)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
PTVXXUDFVRRVAE
|
9.4 | IC50 | 3 | — | |
NRRBFJRUKPITFY
|
9.2 | IC50 | 5 | — | |
ALIRNZFSPVRFPC
|
9.1 | IC50 | 3 | — | |
RUMXSJCIUQZQHF
|
8.7 | IC50 | 3 | — | |
CSXUIGRDFNAIAL
|
8.7 | IC50 | 3 | — | |
MBHHJCMRPHUOAD
|
8.6 | IC50 | 4 | — | |
SPUWUOGLPPVXCW
|
8.5 | IC50 | 15 | Yes | |
LQRGSXMDDSWGQL
|
8.5 | IC50 | 3 | — | |
DLMBMHOJKBPKLK
|
8.5 | IC50 | 5 | — | |
NREVBIQYDIDHPZ
|
8.4 | IC50 | 5 | — | |
XHRZOMIMLIVCLD
|
8.4 | IC50 | 3 | — | |
MKWIGRVAGAAHEM
|
8.3 | IC50 | 3 | — | |
YTSDNPLOCDVGNB
|
8.3 | IC50 | 8 | — | |
KDDHBEBXEUYFNL
|
8.3 | IC50 | 3 | — | |
WZGZBUFREKYIRA
|
8.3 | IC50 | 3 | — | |
PHSBLNQTZKZQLY
|
8.2 | IC50 | 3 | — | |
HEDDQUIXAAICJH
|
8.1 | IC50 | 4 | — | |
BUZYGKOYMBGUKX
|
8.1 | IC50 | 3 | — | |
MMRLNUFECMEMSQ
|
8.1 | IC50 | 3 | — | |
CBWWAMHIIZVQTP
|
8.0 | IC50 | 6 | — | |
SORJWXKYZACWJA
|
8.0 | IC50 | 3 | — | |
MJOCJDMQRCJQJF
|
7.9 | IC50 | 7 | — | |
MZPILEJBIWMIFA
|
7.9 | IC50 | 3 | — | |
CQWRMHYRBJWJNS
|
7.9 | IC50 | 5 | — | |
NMIHFSQPVACNNT
|
7.9 | IC50 | 3 | — | |
XVLBYYUDKFJBBH
|
7.8 | IC50 | 4 | — | |
OROGNMYAIPBPKE
|
7.8 | IC50 | 4 | — | |
HGALDAPNHYJZAJ
|
7.7 | IC50 | 11 | Yes | |
JNIYBOVYGYUEST
|
7.7 | IC50 | 3 | — | |
BBLOBZNVTRKTQL
|
7.5 | IC50 | 5 | — | |
NLZUZMDQCFLSME
|
7.5 | IC50 | 4 | — | |
DKEXUOIKEUTIAL
|
7.5 | IC50 | 3 | — | |
XLHSLEFSSSWIGF
|
7.5 | IC50 | 3 | — | |
BSGWEWBSWAVORO
|
7.3 | IC50 | 5 | — | |
LPHRWFLVTLSQRC
|
7.3 | IC50 | 5 | — | |
DBHCCEYQTJLJOR
|
7.3 | IC50 | 3 | — | |
KKXDIDTZXUDGDY
|
7.3 | IC50 | 4 | — | |
NVFPMSWRLJYMJE
|
7.3 | IC50 | 6 | — | |
OTWGEGUQDHMDBA
|
7.2 | IC50 | 3 | — | |
LTZAOEYIDIFFHJ
|
7.2 | IC50 | 5 | — | |
GZTMFOCEFPOHGW
|
7.2 | IC50 | 5 | — | |
SQZDJBNTERGDSI
|
7.2 | IC50 | 5 | — | |
CXUFYCPSBOYQMV
|
7.1 | IC50 | 5 | — | |
JSONRPFPVGYCOB
|
7.1 | IC50 | 3 | — | |
MILDDBYLPYUFOX
|
7.1 | IC50 | 3 | — | |
SHPLGWYLKVEYNP
|
7.0 | IC50 | 3 | — | |
HGAJCAYHMBFUDT
|
7.0 | IC50 | 3 | — | |
LCQAIZAFSOZWRC
|
7.0 | IC50 | 8 | Yes | |
BERSUAQTWMUYMU
|
7.0 | IC50 | 3 | — | |
OYZYYVWBGXJDCM
|
7.0 | IC50 | 3 | — |