Target Details
| UniProt AC | A3EZJ3 |
|---|---|
| Gene Symbol | NS3 |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 131
- Clinical molecules 0
- Avg pChEMBL 7.09
Active Molecules (131)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
QZYDBDVUQGBCBJ
|
6.5 | Ki | 2 | — | |
YJMIQFUZBHCYMC
|
6.5 | Ki | 2 | — | |
BWWAUBIBIRFGIH
|
6.5 | IC50 | 2 | — | |
DYOHVYXXZTWQRG
|
6.4 | Ki | 2 | — | |
BKFUQKRRUFYLMR
|
6.4 | Ki | 2 | — | |
HZBORGISLFBIJH
|
6.4 | Ki | 2 | — | |
JEUTVNLXGFTXIX
|
6.4 | IC50 | 2 | — | |
BJNLEYZJCBQQNV
|
6.4 | IC50 | 2 | — | |
MXLMCJDWRDDYKD
|
6.4 | Ki | 2 | — | |
YBTIWYVRWNOJDE
|
6.4 | Ki | 2 | — | |
UFWAWGFRBDHWLJ
|
6.4 | IC50 | 2 | — | |
LRQIHHYBLDMHIX
|
6.3 | Ki | 2 | — | |
ZUXXBCGSGVJVMR
|
6.3 | IC50 | 2 | — | |
OFYCIMYEZGXNRV
|
6.3 | IC50 | 2 | — | |
PEMJIWVJFZGEMI
|
6.3 | IC50 | 2 | — | |
LDWPJOSLYTVLDW
|
6.3 | IC50 | 2 | — | |
XICAUTQYHONJLM
|
6.3 | Ki | 2 | — | |
JMQLVAREPUAGLB
|
6.3 | Ki | 2 | — | |
OKRNLCHFEMYBGU
|
6.2 | IC50 | 2 | — | |
AUECKNIWQAGLTA
|
6.2 | IC50 | 2 | — | |
GVJGDZVRCYUEOP
|
6.2 | Ki | 2 | — | |
PHHWHAUDBBQYMR
|
6.2 | Ki | 2 | — | |
OQVXUBNMMPRFKP
|
6.2 | Ki | 2 | — | |
ZEWQUBUPAILYHI
|
6.2 | IC50 | 21 | — | |
UGXJJKIZIYBORF
|
6.2 | IC50 | 2 | — | |
RHMKKGGJMOZLFP
|
6.1 | Ki | 2 | — | |
DXKIEXPGQCEISZ
|
6.1 | Ki | 2 | — | |
YYHBOQQWMBQASJ
|
6.1 | IC50 | 2 | — | |
SDFIBSSAECGDIK
|
6.1 | IC50 | 2 | — | |
JOMMVUMCDVMUOS
|
6.0 | IC50 | 2 | — | |
QHLKHILIWVLAMX
|
6.0 | Ki | 2 | — |