Target Details
| UniProt AC | A3EZI9 |
|---|---|
| Gene Symbol | NS3 |
| Protein Name | Genome polyprotein |
| Organism | Hepacivirus hominis |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF07652 (Flavi_DEAD) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29) |
Summary
- Multi-target molecules 670
- Clinical molecules 0
- Avg pChEMBL 7.83
Active Molecules (670)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
KRVBPGRPHRGDBE
|
9.2 | IC50 | 4 | — | |
ZIHXHTFVLKLWNX
|
9.2 | Ki | 4 | — | |
FVAHUZNNBVVCMP
|
9.2 | Ki | 2 | — | |
RTCPQVJDZHADDP
|
9.2 | Ki | 2 | — | |
YWYUGJWEIJQUGR
|
9.1 | IC50 | 3 | — | |
AGVSXXLDLPSANO
|
9.1 | Ki | 3 | — | |
UDBSCDWKAHTYGU
|
9.1 | Ki | 2 | — | |
DMEMWXCZOKDOMY
|
9.1 | IC50 | 3 | — | |
FTPCVQUWCWXUHD
|
9.1 | IC50 | 2 | — | |
IHPQWLFEUQBMFZ
|
9.1 | IC50 | 4 | — | |
KNQHCQDUNTWSPH
|
9.1 | IC50 | 4 | — | |
LOYIQGBTNJFCIL
|
9.1 | IC50 | 4 | — | |
NVQVBMCNJWRJDK
|
9.1 | Ki | 3 | — | |
OWSMICPTINRUKP
|
9.1 | Ki | 3 | — | |
KUQWGLQLLVFLSM
|
9.0 | Ki | 3 | — | |
LJPHUUAAUHAMGF
|
9.0 | Ki | 3 | — | |
NWFWLEAQCNXLAB
|
9.0 | IC50 | 4 | — | |
NWNRFJLJFPUJSR
|
9.0 | IC50 | 4 | — | |
OIHIJLNMNDCCIY
|
9.0 | IC50 | 4 | — | |
PSVSXONHXYMVQH
|
9.0 | IC50 | 2 | — | |
RZCUJQGMLLHXFG
|
9.0 | IC50 | 4 | — | |
WFXFHGMKTRFARM
|
9.0 | IC50 | 4 | — | |
XRWSZZJLZRKHHD
|
9.0 | IC50 | 3 | — | |
YHJYFWRWHAHNQA
|
9.0 | IC50 | 4 | — | |
XXXWQTLZEUCJPJ
|
8.9 | IC50 | 3 | — | |
BIDQVOKHLFEVMT
|
8.9 | Ki | 3 | — | |
LWPMFURSCCPHJU
|
8.9 | Ki | 3 | — | |
XLLUDKOBZFHIKN
|
8.9 | IC50 | 4 | — | |
WJEOOIPQOGUUDR
|
8.9 | IC50 | 3 | — | |
YUACNGPAVKFBDY
|
8.9 | IC50 | 3 | — | |
DGCPGLRWAMIHKS
|
8.9 | IC50 | 3 | — | |
LKXFEIUKEHYFPB
|
8.9 | Ki | 2 | — | |
MWVCOSKHVKYOCV
|
8.9 | Ki | 3 | — | |
XFYOTNPRWVBFPP
|
8.9 | IC50 | 4 | — | |
MOJHZLPPVIASCY
|
8.8 | IC50 | 4 | — | |
NLCBQIDOYIYGHS
|
8.8 | IC50 | 4 | — | |
PDBMENIRROXLPP
|
8.8 | Ki | 2 | — | |
VXDRIGYTIFAUHJ
|
8.8 | IC50 | 4 | — | |
YNYFVDOGUKBANE
|
8.8 | IC50 | 4 | — | |
AMWXBFDFQCGDLH
|
8.8 | IC50 | 4 | — | |
DMHDFSSOXNVSGH
|
8.8 | Ki | 3 | — | |
GNMJIFOVLJTJGQ
|
8.8 | IC50 | 4 | — | |
LRSKPOKZPAQFRH
|
8.8 | IC50 | 4 | — | |
ORVVZCJIOXCRTD
|
8.8 | Ki | 2 | — | |
VCYVRAYCTRSTDK
|
8.8 | IC50 | 4 | — | |
XJAWIAYPIRGXTP
|
8.8 | Ki | 2 | — | |
NMFUHYFGDLXDAP
|
8.8 | IC50 | 3 | — | |
YQSZHQDSWAVRIF
|
8.8 | IC50 | 3 | — | |
ITOLHHBOXHCVRC
|
8.8 | IC50 | 2 | — | |
WXGVQUUZCZFRQM
|
8.8 | IC50 | 4 | — |