Target Details
UniProt ACA3EZI9
Gene SymbolNS3
Protein NameGenome polyprotein
OrganismHepacivirus hominis
Entry Name
Organism Category Pathogen
Pfam Domains PF07652 (Flavi_DEAD) PF22027 (NS3_helicase_C) PF02907 (Peptidase_S29)
Summary
  • Multi-target molecules 670
  • Clinical molecules 0
  • Avg pChEMBL 7.83
Top Co-occurrence Targets
  • NS4A 647 shared
  • 210 shared
  • NS3/4A 205 shared
  • 49 shared
  • 30 shared
  • 29 shared
  • ELANE 13 shared
  • 10 shared
  • CTRC 9 shared
  • 7 shared
Active Molecules (670)
InChIKey pChEMBL Type Targets Clinical
SRLXXGVPQVHYOH 6.1 Ki 2
JTHOMYNBQBGFIB 6.1 IC50 4
NEAJQBXNBDUFPF 6.1 IC50 4
SSKVGHVPLCLPQX 6.1 IC50 2
PGMJQKKJQFXGPC 6.1 IC50 2
QCINIJBXZXYDNS 6.1 Ki 2
NPAOZMMZEIEAMU 6.1 Ki 2
JMGFJSHONQYBNU 6.1 Ki 3
RDNPNVCQGXONSL 6.1 Ki 2
AQLONSADYDGUDL 6.0 Ki 2
JSLHBHTXPPJVJD 6.0 Ki 2
JWRJMJKIGFHHSI 6.0 Ki 2
KTMGUHOUDWBEQT 6.0 Ki 3
CFWZGBNPCMHIRF 6.0 Ki 2
DRSAXOUTGBMRRP 6.0 Ki 2
JKARAVRHPIXGBJ 6.0 IC50 4
WPCPXTRQGARZPN 6.0 IC50 2
NAHKDQGSUSSLMG 6.0 IC50 2
GSVABYIDKWHKNL 6.0 Ki 2
XQNSGMJILVCEJU 6.0 Ki 3
2D structure