Target Details
| UniProt AC | A0A7G2HKP9 |
|---|---|
| Gene Symbol | N/A |
| Protein Name | Histone deacetylase |
| Organism | Cryptosporidium parvum |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF00850 (Hist_deacetyl) |
Summary
- Multi-target molecules 16
- Clinical molecules 14
- Avg pChEMBL 7.58
Active Molecules (16)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
NXFALCZBQFKESM
|
9.1 | IC50 | 14 | Yes | |
FBOIQKKEKYJGGI
|
9.0 | IC50 | 6 | Yes | |
WMMGXRCXFKMSGF
|
9.0 | IC50 | 14 | Yes | |
CCDVRDJZGFEHAS
|
8.4 | IC50 | 14 | Yes | |
VODSDFCUCFMZGN
|
8.4 | IC50 | 14 | Yes | |
MBUPURNAOZZFIU
|
8.1 | IC50 | 14 | Yes | |
PTHPLNHMLCUQHG
|
8.0 | Ki | 2 | — | |
QCAGJJVUDIGMDW
|
7.5 | IC50 | 14 | Yes | |
SIVWRIUCOPXNRQ
|
7.5 | IC50 | 14 | Yes | |
ZMLFRAJSAWUTBS
|
7.0 | IC50 | 14 | Yes | |
RTKPITSFVVVAGQ
|
6.7 | IC50 | 14 | Yes | |
YHUAYRYAJHEOFC
|
6.7 | IC50 | 14 | Yes | |
YLJIMTMXMYWMMG
|
6.7 | IC50 | 14 | Yes | |
PTHPLNHMLCUQHG
|
6.6 | Ki | 2 | — | |
HLNCULXJFNWYKC
|
6.5 | IC50 | 14 | Yes | |
KKKZOWKRDNZOQP
|
6.1 | IC50 | 14 | Yes |