Target Details
| UniProt AC | A0A1L2E0X0 |
|---|---|
| Gene Symbol | orf1a |
| Protein Name | N/A |
| Organism | Middle East respiratory syndrome-related coronavirus |
| Entry Name | |
| Organism Category | Pathogen |
| Pfam Domains | PF16251 (bCoV_NAB) PF11501 (bCoV_NSP1) PF11633 (bCoV_SUD_M) PF09401 (CoV_NSP10) PF19212 (CoV_NSP2_C) PF19211 (CoV_NSP2_N) PF19218 (CoV_NSP3_C) PF16348 (CoV_NSP4_C) PF19217 (CoV_NSP4_N) PF19213 (CoV_NSP6) PF08716 (CoV_NSP7) PF08717 (CoV_NSP8) PF08710 (CoV_NSP9) PF08715 (CoV_peptidase) PF01661 (Macro) PF05409 (Peptidase_C30) |
Summary
- Multi-target molecules 26
- Clinical molecules 0
- Avg pChEMBL 6.88
Active Molecules (26)
| InChIKey | pChEMBL | Type | Targets | Clinical | |
|---|---|---|---|---|---|
RBBAPAKZARUVHL
|
7.8 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
7.5 | IC50 | 6 | — | |
PAJZPMREBNPURC
|
7.3 | IC50 | 2 | — | |
LPVQTWYXNIFHTH
|
7.3 | IC50 | 2 | — | |
UAFLFCJAOKBHAW
|
7.2 | IC50 | 2 | — | |
MODFCHUDBQIQAH
|
7.2 | IC50 | 2 | — | |
PHUZMTSQHVZDOX
|
7.1 | IC50 | 2 | — | |
BHZBRFONZANPNK
|
7.0 | IC50 | 2 | — | |
XTRGKOYANUJLCC
|
7.0 | IC50 | 2 | — | |
BLRXSZOWSREMKN
|
7.0 | IC50 | 2 | — | |
XXWDDQJFYNJUCB
|
7.0 | IC50 | 3 | — | |
YVCYGQVRUNWVOI
|
7.0 | IC50 | 3 | — | |
FOLCUFKJHSQMEL
|
6.9 | IC50 | 3 | — | |
JAZGKZKQQSCVMM
|
6.8 | IC50 | 2 | — | |
VCQYBHSDNWQLAS
|
6.8 | IC50 | 2 | — | |
WKNCKKOHQQLNCY
|
6.8 | IC50 | 3 | — | |
XCUAIINAJCDIPM
|
6.8 | IC50 | 2 | — | |
NETTVHMSXGRAJR
|
6.8 | IC50 | 2 | — | |
JCBNYZVAMNCKMA
|
6.7 | IC50 | 2 | — | |
TXBSVWQNUSXCIO
|
6.6 | IC50 | 2 | — | |
HWUIYNOFYVRYOP
|
6.5 | IC50 | 2 | — | |
ORKNIPZHPCWIDI
|
6.5 | IC50 | 2 | — | |
AVMDEKFUKVZQPM
|
6.4 | IC50 | 2 | — | |
BSPZFJDYQHDZNR
|
6.4 | IC50 | 7 | — | |
NLVRHQFXQFSBQK
|
6.2 | IC50 | 2 | — | |
PJEUBFINPIVQHS
|
6.2 | IC50 | 2 | — |