Molecule Details
InChIKeyZZZRHFQPNAABMT-QPJJXVBHSA-N
Canonical SMILESCn1cc(-c2ccncc2/C=C/C(=O)Nc2ccc(CN3CC4CC3CO4)cc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24863 CCNC Homo sapiens Human PF16899 PF00134 7.8 IC50 ChEMBL;BindingDB
P49336 CDK8 Homo sapiens Human PF00069 7.8 IC50 ChEMBL