Molecule Details
InChIKeyZZXWQIDOSVIHIM-UHFFFAOYSA-N
Compound Name3-[3-methyl-7-[(1-methylpyrazol-4-yl)methylamino]-1-propan-2-ylpyrazolo[4,5-b]pyridin-5-yl]-1H-pyridin-2-one
Canonical SMILESCc1nn(C(C)C)c2c(NCc3cnn(C)c3)cc(-c3ccc[nH]c3=O)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.11
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q01064 PDE1B Homo sapiens Human PF00233 PF08499 7.7 IC50 ChEMBL;BindingDB
P54750 PDE1A Homo sapiens Human PF00233 PF08499 6.9 IC50 ChEMBL;BindingDB
Q14123 PDE1C Homo sapiens Human PF00233 PF08499 6.7 IC50 ChEMBL;BindingDB