Molecule Details
InChIKeyZZIYTDPDYPNEHS-UHFFFAOYSA-N
Compound Name1-[3-[[4,4-Dimethyl-8-(propan-2-ylamino)-11-oxa-9,14,16-triazatetracyclo[8.7.0.02,7.012,17]heptadeca-1(10),2(7),8,12(17),13,15-hexaen-13-yl]amino]propyl]pyrrolidin-2-one
Canonical SMILESCC(C)Nc1nc2oc3c(NCCCN4CCCC4=O)ncnc3c2c2c1CCC(C)(C)C2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07343 PDE4B Homo sapiens Human PF18100 PF00233 10.0 IC50 ChEMBL;BindingDB
Q08499 PDE4D Homo sapiens Human PF18100 PF00233 10.0 IC50 ChEMBL;BindingDB
P27815 PDE4A Homo sapiens Human PF18100 PF00233 9.5 IC50 ChEMBL;BindingDB