Molecule Details
InChIKeyZZFYPMWQKLOJIR-MRXNPFEDSA-N
Compound Name(2R)-2-[1,1-dioxo-7-(4-phenylphenoxy)-4,5-dihydro-3H-1lambda6,2,5-benzothiadiazepin-2-yl]-N-hydroxypropanamide
Canonical SMILESC[C@H](C(=O)NO)N1CCNc2cc(Oc3ccc(-c4ccccc4)cc3)ccc2S1(=O)=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.59
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 8.6 pIC50 TTD_MultiTarget
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.6 pIC50 TTD_MultiTarget