Molecule Details
InChIKeyZZCZGLYROGNMLJ-UHFFFAOYSA-N
Compound Name4-[1-[3-[(2,2-Difluorocyclopropanecarbonyl)amino]phenyl]propylamino]quinazoline-8-carboxamide
Canonical SMILESCCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)C2CC2(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 9.3 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.6 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.9 IC50 ChEMBL;BindingDB