Molecule Details
InChIKeyZYXGKENMDDPQIE-UHFFFAOYSA-N
Compound Name2-(furan-2-yl)-N-[(4-methoxyphenyl)methyl]-5-(methylamino)-[1,2,4]triazolo[1,5-c]pyrimidine-8-carboxamide
Canonical SMILESCNc1ncc(C(=O)NCc2ccc(OC)cc2)c2nc(-c3ccco3)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.46
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0DMS8 ADORA3 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.1 Ki ChEMBL;BindingDB