Molecule Details
InChIKeyZYWJPJYYTUCZHN-UHFFFAOYSA-N
Compound NameN-ethyl-4-(4-(2-phenyl-1H-indol-3-yl)pyrimidin-2-ylamino)piperidine-1-carboxamide
Canonical SMILESCCNC(=O)N1CCC(Nc2nccc(-c3c(-c4ccccc4)[nH]c4ccccc34)n2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.09
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 8.3 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.7 IC50 ChEMBL;BindingDB