Molecule Details
InChIKeyZYPJRFNOUPSZFL-UHFFFAOYSA-N
Compound NameN-(3,4-dichlorobenzyl)-2-(1H-indazol-5-yl)pyrimidin-4-amine
Canonical SMILESClc1ccc(CNc2ccnc(-c3ccc4[nH]ncc4c3)n2)cc1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49760 CLK2 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
Q9HAZ1 CLK4 Homo sapiens Human PF00069 6.6 IC50 ChEMBL;BindingDB
Q9Y463 DYRK1B Homo sapiens Human PF00069 6.3 IC50 ChEMBL;BindingDB