Molecule Details
InChIKeyZYLHCSSOEGIFAO-UHFFFAOYSA-N
Compound NameN-[3-({4-[(3-Aminopropyl)amino]-5-Iodopyrimidin-2-Yl}amino)phenyl]pyrrolidine-1-Carboxamide
Canonical SMILESNCCCNc1nc(Nc2cccc(NC(=O)N3CCCC3)c2)ncc1I
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.5
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75385 ULK1 Homo sapiens Human PF12063 PF21127 PF00069 6.9 IC50 ChEMBL;BindingDB
Q8IYT8 ULK2 Homo sapiens Human PF12063 PF21127 PF00069 6.4 IC50 ChEMBL;BindingDB
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 6.2 IC50 ChEMBL;BindingDB