Molecule Details
InChIKeyZXXCWRYARSIMPM-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(CCOC(c2ccc(Cl)cc2)(c2ccc(Cl)cc2)C(Oc2nc3c(c(OC)n2)CCC3)C(=O)O)cc1OC
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 6.7 Ki ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB