Molecule Details
InChIKeyZXRLFIJLBNQELO-UHFFFAOYSA-N
Compound NameN'-(4H-1,3-benzodioxin-6-yl)-4-(6-bromo-13-chloro-4-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-ylidene)-N-cyanopiperidine-1-carboximidamide
Canonical SMILESN#CN/C(=N/c1ccc2c(c1)COCO2)N1CCC(=C2c3ccc(Cl)cc3CCc3cc(Br)cnc32)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.82
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.8 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.8 IC50 ChEMBL