Molecule Details
InChIKeyZWYOUKDNWVHYPO-BGLQLSEMSA-N
Compound Name(1R,4S,9aR,11aR)-6-ethyl-4,9a,11a-trimethyl-1-(6-methylheptan-2-yl)-2,3,3a,3b,4,5,5a,8,9,9b,10,11-dodecahydro-1H-indeno[5,4-f]quinolin-7-one
Canonical SMILESCCN1C(=O)CC[C@]2(C)C3CC[C@@]4(C)C(CC[C@@H]4C(C)CCCC(C)C)C3[C@@H](C)CC12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.48
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18405 SRD5A1 Homo sapiens Human PF02544 8.5 IC50 ChEMBL;BindingDB
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 8.5 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 8.5 pIC50 TTD_MultiTarget