Molecule Details
InChIKeyZWSQJIRFQBKTDD-GLDPKNIUSA-N
Compound Name(2S)-2-[[(2S,3aS,6R,7aS)-6-hydroxy-1-[(2R)-2-[[(2R)-2-hydroxy-3-(4-hydroxyphenyl)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]-2,3,3a,4,5,6,7,7a-octahydroindole-2-carbonyl]amino]-5-(diaminomethylideneamino)pentanoic acid
Canonical SMILESN=C(N)NCCC[C@H](NC(=O)[C@@H]1C[C@@H]2CC[C@@H](O)C[C@@H]2N1C(=O)[C@@H](Cc1ccc(O)cc1)NC(=O)[C@H](O)Cc1ccc(O)cc1)C(=O)O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P07477 PRSS1 Homo sapiens Human PF00089 6.0 IC50 ChEMBL;BindingDB
P07478 PRSS2 Homo sapiens Human PF00089 6.0 IC50 ChEMBL
P35030 PRSS3 Homo sapiens Human PF00089 6.0 IC50 ChEMBL