Molecule Details
InChIKeyZWSIFNIMWCIVIU-FTYNLOLUSA-N
Compound NameH-Gly-Cys-Cys-Ser-Leu-Pro-Pro-Cys-Ala-Leu-Ser-Asn-Pro-Asp-Tyr-Cys-NH2
Canonical SMILESCC(C)C[C@H](NC(=O)[C@H](C)NC(=O)[C@H](CS)NC(=O)[C@@H]1CCCN1C(=O)[C@@H]1CCCN1C(=O)[C@H](CC(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CS)NC(=O)[C@H](CS)NC(=O)CN)C(=O)N[C@@H](CO)C(=O)N[C@@H](CC(N)=O)C(=O)N1CCC[C@H]1C(=O)N[C@@H](CC(=O)O)C(=O)N[C@@H](Cc1ccc(O)cc1)C(=O)N[C@@H](CS)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P17787 CHRNB2 Homo sapiens Human PF02931 PF02932 7.2 IC50 ChEMBL;BindingDB
P32297 CHRNA3 Homo sapiens Human PF02931 PF02932 7.2 IC50 ChEMBL
P36544 CHRNA7 Homo sapiens Human PF02931 PF02932 7.2 IC50 ChEMBL;BindingDB