Molecule Details
InChIKeyZWRLLBAFCKACAL-UHFFFAOYSA-N
Compound Name8-[[4-(Aminocarbonyl)-2-methoxyphenyl]amino]-N-(2,6-diethylphenyl)-4,5-dihydro-1-methyl-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide
Canonical SMILESCCc1cccc(CC)c1NC(=O)c1nn(C)c2c1CCc1cnc(Nc3ccc(C(N)=O)cc3OC)nc1-2
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.56
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33981 TTK Homo sapiens Human PF00069 7.4 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 6.1 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.1 pIC50 TTD_MultiTarget