Molecule Details
InChIKeyZWNFGXDUPNOZMG-UHFFFAOYSA-N
Compound Name5-(N-[cyclopentanecarbonyl]amino)-3-(1-methylpiperidin-4-yl)pyrrolo[3,2-b]pyridine
Canonical SMILESCN1CCC(c2c[nH]c3ccc(NC(=O)C4CCCC4)nc23)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.76
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P30939 HTR1F Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.2 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB