Molecule Details
InChIKeyZWLPFMJOMZEBOD-UHFFFAOYSA-N
Compound Name1-(4-(3-amino-7-((4-methylpiperazin-1-yl)methyl)-1H-indazol-4-yl)phenyl)-3-m-tolylurea
Canonical SMILESCc1cccc(NC(=O)Nc2ccc(-c3ccc(CN4CCN(C)CC4)c4[nH]nc(N)c34)cc2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.63
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P36888 FLT3 Homo sapiens Human PF00047 PF07714 6.7 IC50 ChEMBL;BindingDB
Q02161 RHD Homo sapiens Human PF00909 6.7 pIC50 TTD_MultiTarget
P10721 KIT Homo sapiens Human PF00047 PF07714 6.5 IC50 ChEMBL;BindingDB