Molecule Details
InChIKeyZWBIIYBHVNHQOG-UHFFFAOYSA-N
Compound Name1-[2-(1,3-Dihydroisoindol-2-yl)ethyl]-3-[3-(trifluoromethoxy)phenyl]imidazolidin-2-one
Canonical SMILESO=C1N(CCN2Cc3ccccc3C2)CCN1c1cccc(OC(F)(F)F)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35462 DRD3 Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P14416 DRD2 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.2 IC50 ChEMBL;BindingDB