Molecule Details
InChIKeyZVVCSBSDFGYRCB-UHFFFAOYSA-N
Canonical SMILESCCCc1c(OCCCOc2ccc(C(C)=O)c(OC)c2CCC)ccc2c1OC(C(=O)O)CC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB17101
Drug NameSC 41930
CAS Number120072-59-5
Groups experimental
ATC Codes nan
Descriptionnan

Categories: Analgesics Analgesics, Non-Narcotic Anti-Inflammatory Agents Anti-Inflammatory Agents, Non-Steroidal Antirheumatic Agents Heterocyclic Compounds, Fused-Ring Hormone Antagonists Hormones, Hormone Substitutes, and Hormone Antagonists Leukotriene Antagonists Peripheral Nervous System Agents Pyrans Sensory System Agents
Cross-references: BindingDB: 50001610 CHEMBL14823 ChemSpider: 102927
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NPC1 LTB4R2 Homo sapiens Human PF00001 7.0 Ki ChEMBL;BindingDB
Q15722 LTB4R Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
DrugBank Target Actions (2)
Target Gene Target Name Action Type
Q15722 LTB4R Leukotriene B4 receptor 1 binder targets
Q9NPC1 LTB4R2 Leukotriene B4 receptor 2 inhibitor targets