Molecule Details
InChIKeyZVTDLPBHTSMEJZ-JSZLBQEHSA-N
Compound NameDanoprevir
Canonical SMILESCC(C)(C)OC(=O)N[C@H]1CCCCC/C=C\[C@@H]2C[C@@]2(C(=O)NS(=O)(=O)C2CC2)NC(=O)[C@@H]2C[C@@H](OC(=O)N3Cc4cccc(F)c4C3)CN2C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB11779
Drug NameDanoprevir
CAS Number850876-88-9
Groups investigational
ATC Codes nan
DescriptionDanoprevir has been used in trials studying the treatment of Hepatitis C, Chronic.

Categories: Amides Amino Acids Amino Acids, Cyclic Amino Acids, Peptides, and Proteins Cycloparaffins Cytochrome P-450 CYP3A Inhibitors Cytochrome P-450 CYP3A4 Inhibitors Cytochrome P-450 CYP3A4 Inhibitors (strong) Cytochrome P-450 Enzyme Inhibitors Heterocyclic Compounds, Fused-Ring Imino Acids Lactams Sulfones Sulfur Compounds
Cross-references: CHEMBL258734 ChemSpider: 9460579 PubChem:11285588 PubChem:347828129 Wikipedia: Danoprevir ZINC: ZINC000029058869
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
A3EZI9 NS3 Hepacivirus hominis Pathogen PF07652 PF22027 PF02907 9.7 IC50 ChEMBL;BindingDB
D2K2A8 NS4A Hepacivirus hominis Pathogen PF01006 9.7 IC50 ChEMBL
F5B4I0 Hepacivirus hominis Pathogen PF01001 9.7 IC50 ChEMBL
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P08684 CYP3A4 Cytochrome P450 3A4 inhibitor enzymes
P26664 Genome polyprotein binder targets
P03366 gag-pol Gag-Pol polyprotein inhibitor targets