Molecule Details
InChIKeyZVKJUDYDWABBFR-UHFFFAOYSA-N
Compound Name2''-(1-Methyl-1H-pyrazol-3-ylamino)-6-piperazin-1-yl[2,4'']bipyridinyl-4-carbonitrile
Canonical SMILESCn1ccc(Nc2cc(-c3cc(C#N)cc(N4CCNCC4)n3)ccn2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.48
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15139 PRKD1 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 8.1 IC50 ChEMBL;BindingDB
Q13563 PKD2 Homo sapiens Human PF18109 PF08016 PF20519 7.2 IC50 BindingDB
Q9BZL6 PRKD2 Homo sapiens Human PF00130 PF00169 PF00069 PF25525 7.2 IC50 ChEMBL