Molecule Details
InChIKeyZUTFDMVDCHXOFA-UHFFFAOYSA-N
Compound Name3-Chloro-2'-Cyano-5'-(1h-1,2,4-Triazol-1-Ylmethyl)biphenyl-4-Yl Sulfamate
Canonical SMILESN#Cc1ccc(Cn2cncn2)cc1-c1ccc(OS(N)(=O)=O)c(Cl)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.21
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11511 CYP19A1 Homo sapiens Human PF00067 9.3 IC50 ChEMBL;BindingDB
P08842 STS Homo sapiens Human PF00884 PF14707 8.3 IC50 ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 7.1 IC50 ChEMBL;BindingDB