Molecule Details
InChIKeyZTEDLCUEUUWRAT-UHFFFAOYSA-N
Compound NameN,6-dimethyl-5-[4-[(4-oxo-5H-furo[3,2-c]quinolin-7-yl)methyl]piperazin-1-yl]pyridine-2-carboxamide
Canonical SMILESCNC(=O)c1ccc(N2CCN(Cc3ccc4c(c3)[nH]c(=O)c3ccoc34)CC2)c(C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.39
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P09874 PARP1 Homo sapiens Human PF00533 PF21728 PF00644 PF02877 PF05406 PF00645 PF08063 9.2 IC50 BindingDB
Q9UGN5 PARP2 Homo sapiens Human PF00644 PF02877 PF05406 6.8 IC50 BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.2 IC50 BindingDB