Molecule Details
InChIKeyZSGSJOKPFNUESJ-UHFFFAOYSA-N
Compound Name2,2,2-Trifluoro-1-(5-(4-(5-phenyl-1,3,4-oxadiazol-2-yl)piperidine-1-carbonyl)thiophen-2-yl)ethanone
Canonical SMILESO=C(c1ccc(C(=O)C(F)(F)F)s1)N1CCC(c2nnc(-c3ccccc3)o2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.8
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q02161 RHD Homo sapiens Human PF00909 6.8 pIC50 TTD_MultiTarget
Q13547 HDAC1 Homo sapiens Human PF00850 6.8 pIC50 TTD_MultiTarget
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.8 IC50 ChEMBL;BindingDB