Molecule Details
InChIKeyZSBXISJADFDHQV-UHFFFAOYSA-N
Compound Name(1-Methylsulfonylindol-5-yl)-[3-([1,2,4]triazolo[1,5-a]pyrimidin-7-yl)piperidin-1-yl]methanone
Canonical SMILESCS(=O)(=O)n1ccc2cc(C(=O)N3CCCC(c4ccnc5ncnn45)C3)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O00408 PDE2A Homo sapiens Human PF01590 PF00233 8.6 IC50 ChEMBL;BindingDB
Q14432 PDE3A Homo sapiens Human PF00233 6.1 IC50 ChEMBL;BindingDB